SCHEMBL8570512

SCHEMBL8570512

c1ccc([C@@H]2CNc3ccccc3C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.51
DAPK3 O43293 1/20 0.42
JAK2 O60674 1/20 0.42
CSF1R P07333 1/20 0.42
RET P07949 1/20 0.42
PRKACA P17612 1/20 0.42
LTK P29376 1/20 0.42
GRK5 P34947 1/20 0.42
KDR P35968 1/20 0.42
MAP2K2 P36507 1/20 0.42
MAPK8 P45983 1/20 0.42
CSNK1A1 P48729 1/20 0.42
CDK8 P49336 1/20 0.42
CLK2 P49760 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
CDK9 P50750 1/20 0.42
RPS6KA3 P51812 1/20 0.42
LIMK1 P53667 1/20 0.42
CDK5 Q00535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570515 1.00 ESR2 (0.51) ESR2DAPK3JAK2CSF1RRET
SCHEMBL29746181 1.00 ESR2 (0.51) ESR2DAPK3JAK2CSF1RRET
SCHEMBL8570510 1.00 ESR2 (0.51) ESR2DAPK3JAK2CSF1RRET
SCHEMBL2361951 0.87 CYP19A1 (0.51) ESR2DAPK3JAK2CSF1RRET
SCHEMBL2362933 0.86 ESR2 (0.50) ESR2MTNR1AMTNR1BMEN1KMT2A
SCHEMBL10536101 0.86 ESR2 (0.50) ESR2MTNR1AMTNR1BMEN1KMT2A
SCHEMBL26613583 0.83 CYP11B2 (0.47) ESR2MEN1KMT2AMAPTCYP2D6
SCHEMBL29746385 0.83 CYP11B2 (0.47) ESR2MEN1KMT2AMAPTCYP2D6
SCHEMBL17634083 0.82 ESR2 (0.47) ESR2MEN1KMT2AGAAMAPT
SCHEMBL29746277 0.82 ESR2 (0.50) ESR2JAK2MTNR1AMTNR1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed