SCHEMBL8570870

SCHEMBL8570870

COc1ccc(S(=O)(=O)Nc2cc(C(=O)CCCCCl)c(OC)cc2OC)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.61
HTR2B P41595 12/20 0.61
HTR2A P28223 8/20 0.61
ALDH1A1 P00352 2/20 0.53
MAPT P10636 2/20 0.53
MAPK1 P28482 2/20 0.53
ALOX15 P16050 2/20 0.53
HSD17B10 Q99714 1/20 0.53
LMNA P02545 3/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 2/20 0.51
HTT P42858 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
KMT2A Q03164 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MEN1 O00255 2/20 0.49
CYP3A4 P08684 1/20 0.49
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8573905 0.92 HTR2C (0.62) HTR2CHTR2BHTR2AALDH1A1MAPK1
SCHEMBL8567723 0.92 HTR2C (0.62) HTR2CHTR2BHTR2AALDH1A1ALOX15
SCHEMBL8572332 0.91 HTR2C (0.53) HTR2CHTR2BHTR2AALDH1A1MAPK1
SCHEMBL8574314 0.90 HTR2C (0.60) HTR2CHTR2BHTR2AALDH1A1MAPT
SCHEMBL8573974 0.90 HTR2C (0.64) HTR2CHTR2BHTR2AALDH1A1MAPK1
SCHEMBL8574255 0.89 HTR2C (0.62) HTR2CHTR2BHTR2AALDH1A1MAPT
SCHEMBL8569901 0.89 HTR2C (0.62) HTR2CHTR2BHTR2AALDH1A1MAPK1
SCHEMBL8811616 0.88 HTR2C (0.63) HTR2CHTR2BHTR2AALDH1A1MAPT
SCHEMBL8570844 0.88 HTR2C (0.63) HTR2CHTR2BHTR2AALDH1A1MAPK1
SCHEMBL8571173 0.88 POLB (0.51) HTR2CHTR2BHTR2AALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed