SCHEMBL8574602

SCHEMBL8574602

C=CCc1c(-c2cc(=O)c3c(O)c(CC=C)c(OCC4=COC(C)(C)O4)cc3o2)ccc(OC)c1OC(C=O)OCC

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 2/20 0.34
MAPT P10636 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP1A1 P04798 2/20 0.33
CYP1B1 Q16678 2/20 0.33
AKT1 P31749 1/20 0.33
CYP1A2 P05177 1/20 0.33
OPRD1 P41143 1/20 0.33
FLT3 P36888 2/20 0.33
AURKA O14965 1/20 0.33
KDR P35968 1/20 0.33
AURKB Q96GD4 1/20 0.33
SOAT2 O75908 1/20 0.33
QPCT Q16769 1/20 0.33
CREB1 P16220 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306598 0.86 AKT1 (0.40) PTGS1PTGS2KDM4EPOLBMAPT
SCHEMBL8427197 0.85 PTGS1 (0.36) PTGS1PTGS2KDM4EPOLBMAPT
SCHEMBL8572731 0.84 QPCT (0.38) POLBMAPTADORA3CYP1A1CYP1B1
SCHEMBL8431327 0.81 KDM4E (0.38) PTGS1PTGS2KDM4EPOLBMAPT
SCHEMBL8309735 0.79 KDM4E (0.39) KDM4EPOLBMAPTADORA3CYP1A1
SCHEMBL8574605 0.78 PTGS1 (0.34) PTGS1PTGS2KDM4EPOLBMAPT
SCHEMBL8308992 0.77 MAOB (0.39) KDM4EPOLBMAPTADORA3CYP1A1
SCHEMBL8310185 0.77 MAOB (0.41) KDM4EPOLBMAPTADORA3CYP1A1
SCHEMBL8306988 0.77 CYP1B1 (0.42) POLBMAPTCYP1A1CYP1B1CYP1A2
SCHEMBL8306599 0.75 FLT3 (0.47) KDM4EPOLBMAPTADORA3CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792789-A TREATING HYPERPERMEABILITY AND INFLAMMATION ADIR ET COMPAGNIE (FR) 1998-08-11 US disclosed