SCHEMBL8576451

SCHEMBL8576451

COc1cc(O)c2c(=O)c(-c3cccc(Cl)c3)cn(C)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 1.00
ABL1 P00519 1/20 0.46
ABL2 P42684 1/20 0.46
SRC P12931 1/20 0.46
GSK3B P49841 3/20 0.44
PRKCA P17252 2/20 0.44
BRD4 O60885 1/20 0.42
NPC1 O15118 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MAPT P10636 2/20 0.40
ABCB1 P08183 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579701 0.86 EGFR (0.79) EGFRABL1ABL2SRCBRD4
SCHEMBL8575324 0.86 EGFR (0.75) EGFRABL1ABL2SRCNPC1
SCHEMBL8572765 0.86 EGFR (0.75) EGFRABL1ABL2SRCNPC1
SCHEMBL8577298 0.86 EGFR (0.78) EGFRABL1ABL2SRCNPC1
SCHEMBL7256796 0.83 EGFR (0.71) EGFRNPC1CYP2C9CYP2C19MAPT
SCHEMBL8575444 0.83 EGFR (0.84) EGFRABL1ABL2SRCNPC1
SCHEMBL8574540 0.83 EGFR (1.00) EGFRABL1ABL2SRCNPC1
SCHEMBL8577489 0.82 EGFR (0.70) EGFRABL1ABL2SRCNPC1
SCHEMBL8601752 0.82 EGFR (1.00) EGFRABL1ABL2SRCMAPT
SCHEMBL8576546 0.82 EGFR (0.82) EGFRABL1ABL2SRCNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO claimed
WO-1998017662-A1 PHENYL-SUBSTITUTED BICYCLIC HETEROCYCLYL DERIVATIVES AND THEIR USE NOVARTIS AG (CH) 1998-04-30 WO disclosed