SCHEMBL8576502

SCHEMBL8576502

CCCOCC[C@H]1CN(C(=O)c2cccc3cccnc23)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.50
POLB P06746 2/20 0.44
KDM4E B2RXH2 1/20 0.42
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
FNTA P49354 6/20 0.40
FNTB P49356 6/20 0.40
MGLL Q99685 1/20 0.37
CCR3 P51677 2/20 0.37
CXCR3 P49682 3/20 0.36
CHRM2 P08172 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8573446 0.91 PARP1 (0.52) PARP1POLBKDM4EHCRTR1HCRTR2
SCHEMBL8573445 0.91 PARP1 (0.52) PARP1POLBKDM4EHCRTR1HCRTR2
SCHEMBL8578507 0.89 PARP1 (0.51) PARP1POLBKDM4EHCRTR1HCRTR2
SCHEMBL8578509 0.89 PARP1 (0.51) PARP1POLBKDM4EHCRTR1HCRTR2
SCHEMBL8574801 0.86 FNTA (0.51) PARP1POLBFNTAFNTBALDH1A1
SCHEMBL6056523 0.78 FNTA (0.62) HCRTR1HCRTR2HTR2AHTR2CFNTA
Hydrochloric Acid SCHEMBL9214284 0.77 FNTA (0.62) HCRTR1HCRTR2HTR2AHTR2CFNTA
SCHEMBL8453359 0.77 FNTA (0.59) PARP1POLBFNTAFNTBALDH1A1
SCHEMBL8453364 0.77 FNTA (0.59) PARP1POLBFNTAFNTBALDH1A1
SCHEMBL8576156 0.77 FNTA (0.51) PARP1FNTAFNTBMGLLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736539-A ANITCARCINOGENIC AGENTS MERCK & CO., INC. (US) 1998-04-07 US disclosed
WO-1995000497-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1995-01-05 WO disclosed