SCHEMBL8577296

SCHEMBL8577296

O=C(NCc1ccc(Nc2n[nH]c3ncnc(Nc4cccc(Cl)c4)c23)cc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.68
ABL1 P00519 8/20 0.68
CDK1 P06493 7/20 0.68
PRKCA P17252 4/20 0.68
SRC P12931 5/20 0.61
ABL2 P42684 1/20 0.48
MT-CO2 P00403 1/20 0.47
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
CNR2 P34972 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6186191 0.89 EGFR (0.67) EGFRABL1CDK1PRKCASRC
SCHEMBL8122065 0.88 EGFR (0.66) EGFRABL1CDK1PRKCASRC
SCHEMBL6189215 0.86 EGFR (0.64) EGFRABL1CDK1PRKCASRC
SCHEMBL8577275 0.86 EGFR (0.63) EGFRABL1CDK1PRKCASRC
SCHEMBL6190120 0.85 EGFR (0.62) EGFRABL1CDK1PRKCASRC
SCHEMBL6184979 0.85 EGFR (0.62) EGFRABL1CDK1PRKCASRC
SCHEMBL6190406 0.85 EGFR (0.67) EGFRABL1CDK1PRKCASRC
SCHEMBL6187136 0.85 EGFR (0.61) EGFRABL1CDK1PRKCASRC
SCHEMBL6187995 0.85 EGFR (0.66) EGFRABL1CDK1PRKCASRC
SCHEMBL6187645 0.84 EGFR (0.66) EGFRABL1CDK1PRKCASRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998014449-A1 FUSED PYRAZOLE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1998-04-09 WO claimed