SCHEMBL8577964

SCHEMBL8577964

COc1ccc(CCn2c(N)c(NC(=O)C3CCCC3)c(=O)[nH]c2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
MAPT P10636 4/20 0.43
G6PD P11413 3/20 0.43
NPC1 O15118 1/20 0.43
MAPK1 P28482 1/20 0.43
P2RX7 Q99572 1/20 0.43
DAO P14920 1/20 0.43
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 5/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 1/20 0.41
RECQL P46063 1/20 0.41
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8575326 0.90 TSHR (0.49) KDM4EMAPTNPC1P2RX7TP53
SCHEMBL8577820 0.87 HTT (0.43) KDM4EMAPTMAPK1DAOTP53
SCHEMBL8576994 0.81 MEN1 (0.52) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL8579589 0.80 KMT2A (0.45) KDM4EKMT2AMEN1ALDH1A1
SCHEMBL8577000 0.76 MEN1 (0.47) KDM4EMAPTNPC1P2RX7TP53
SCHEMBL8579118 0.75 DAO (0.58) KDM4EMAPTG6PDNPC1MAPK1
SCHEMBL8576798 0.71 DAO (0.53) KDM4EMAPTG6PDNPC1MAPK1
SCHEMBL9402327 0.70 ADORA2A (0.44) KDM4EMAPTNPC1TP53RAB9A
SCHEMBL8577647 0.69 DAO (0.52) KDM4EMAPTG6PDNPC1MAPK1
SCHEMBL8579120 0.67 ADORA1 (0.64) KDM4EMAPTG6PDNPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed