SCHEMBL8577647

SCHEMBL8577647

COc1ccc(CCCn2c(N)c(N)c(=O)[nH]c2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.52
LMNA P02545 1/20 0.51
MAPT P10636 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
G6PD P11413 1/20 0.46
MAPK1 P28482 1/20 0.46
HPGD P15428 1/20 0.46
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 4/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 3/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
MEN1 O00255 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579118 0.92 DAO (0.58) DAOMAPTKDM4ENPC1G6PD
SCHEMBL8581809 0.85 DAO (0.48) DAOLMNAMAPTKDM4ENPC1
SCHEMBL6093318 0.84 ALDH1A1 (0.56) DAOMAPTKDM4EMAPK1HPGD
SCHEMBL8576806 0.80 KMT2A (0.59) DAOLMNAMAPTKDM4ENPC1
SCHEMBL8576798 0.78 DAO (0.53) DAOLMNAMAPTKDM4ENPC1
SCHEMBL8579776 0.75 MAPT (0.49) LMNAMAPTKDM4EALDH1A1KMT2A
SCHEMBL1947719 0.75 KMT2A (0.59) DAOLMNAMAPTKDM4ENPC1
SCHEMBL9412486 0.74 ALDH1A1 (0.51) DAOMAPTKDM4ENPC1G6PD
SCHEMBL8581796 0.74 DAO (0.55) DAOLMNAKDM4EHPGDALDH1A1
SCHEMBL8576934 0.74 L3MBTL1 (0.44) DAOLMNAMAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
EP-0654033-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1995-05-24 EP disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed