SCHEMBL8580776

SCHEMBL8580776

COC(=O)CC(NO)C(=O)OC

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
MGAM O43451 2/20 0.37
GAA P10253 2/20 0.37
SI P14410 2/20 0.37
MGAM2 Q2M2H8 2/20 0.37
HSD17B10 Q99714 1/20 0.37
BIRC2 Q13490 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KMT2A Q03164 2/20 0.32
TET2 Q6N021 1/20 0.31
CA14 Q9ULX7 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8580782 1.00 TSHR (0.40) TSHRCA1CA2CA12CA9
SCHEMBL20022609 0.84 TSHR (0.42) TSHRCA1CA2CA12CA9
SCHEMBL13033614 0.82 TSHR (0.40) TSHRCA1CA2CA12CA9
SCHEMBL1891853 0.82 TSHR (0.40) TSHRCA1CA2CA12CA9
SCHEMBL28625413 0.82 TSHR (0.40) TSHRCA1CA2CA12CA9
SCHEMBL27992708 0.80 CA1 (0.40) TSHRCA1CA2CA12CA9
SCHEMBL27992709 0.80 CA1 (0.40) TSHRCA1CA2CA12CA9
SCHEMBL14097419 0.80 CA12 (0.40) TSHRCA1CA2CA12CA9
SCHEMBL19090744 0.80 TSHR (0.39) TSHRCA1CA2CA12CA9
SCHEMBL19670133 0.80 CA12 (0.40) TSHRCA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US claimed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US claimed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP claimed
CN-1058205-A The method for preparing pyridine and quinoline HOECHST CELANESE CORP (US) 1992-01-29 CN claimed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP claimed
US-5808067-A Process for preparing pyridine and quinoline derivatives HOECHST CELANESE CORPORATION (US) 1998-09-15 US disclosed
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US disclosed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US disclosed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP disclosed
CN-1058205-A The method for preparing pyridine and quinoline HOECHST CELANESE CORP (US) 1992-01-29 CN disclosed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP disclosed