SCHEMBL8583397

SCHEMBL8583397

CCN(O)[C@@](CC)(CC(=O)O)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
ALDH1A1 P00352 3/20 0.34
HMGCR P04035 1/20 0.34
CHRM1 P11229 1/20 0.34
TBXA2R P21731 1/20 0.34
ADRA1A P35348 1/20 0.34
KDM4E B2RXH2 3/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
MEN1 O00255 2/20 0.31
CYP1A2 P05177 2/20 0.31
KMT2A Q03164 2/20 0.31
THRB P10828 1/20 0.31
FFAR3 O14843 1/20 0.31
FFAR1 O14842 1/20 0.30
CPT2 P23786 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4998501 0.77 CYP2D6 (0.39) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL9709625 0.77
SCHEMBL29084381 0.76 TSHR (0.35) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL1173130 0.76 TSHR (0.35) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL13276122 0.74 TDP1 (0.33) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL9279731 0.72 ALDH1A1 (0.33) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL28885649 0.72 FFAR3 (0.35) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL8583429 0.71 CYP2D6 (0.34) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL6562033 0.70 TSHR (0.36) TSHRCYP2D6CYP2C19HIF1AALDH1A1
SCHEMBL18798914 0.69 ALDH1A1 (0.46) TSHRCYP2D6CYP2C19HIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US claimed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US claimed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP claimed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP claimed
EP-0415767-A2 Process for preparing pyridine carboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-03-06 EP claimed
US-5808067-A Process for preparing pyridine and quinoline derivatives HOECHST CELANESE CORPORATION (US) 1998-09-15 US disclosed
US-5405987-A N-hydroxyaspartic acid derivatives; chemical intermediates HOECHST CELANESE CORPORATION (US) 1995-04-11 US disclosed
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US disclosed
EP-0564083-A1 Conversion of pyridine-2,3-dicarboxylic acid esters to their cyclic anhydrides HOECHST CELANESE CORPORATION (US) 1993-10-06 EP disclosed
US-5208342-A Hydrolysis and dehydration HOECHST CELANESE CORPORATION (US) 1993-05-04 US disclosed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP disclosed
EP-0452094-A2 A method of the preparation of N-hydroxy aspartic acid derivate HOECHST CELANESE CORPORATION (US) 1991-10-16 EP disclosed
EP-0415767-A2 Process for preparing pyridine carboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-03-06 EP disclosed