SCHEMBL8585044

SCHEMBL8585044

CSc1ccc(O[C@@H]2C[C@H]3[C@@H]4CCC[C@@]4(C)CC[C@@H]3[C@@]3(C)CCCC[C@H]23)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
NR1I3 Q14994 1/20 0.36
GRIN1 Q05586 5/20 0.35
GRIN2B Q13224 5/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
STS P08842 2/20 0.33
EPHX2 P34913 1/20 0.33
CYP19A1 P11511 3/20 0.31
SHBG P04278 1/20 0.31
MBOAT4 Q96T53 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8585049 1.00 CDK5 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8586469 0.87 CDK5 (0.37) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8586472 0.87 CDK5 (0.37) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8582194 0.83 GRIN1 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8582196 0.83 GRIN1 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8585577 0.79 GRIN1 (0.43) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8585574 0.79 GRIN1 (0.43) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8586439 0.73 CDK5 (0.45) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8586432 0.73 CDK5 (0.45) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8334768 0.72 CDK5 (0.35) CDK5CDK5R1NR1I3GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP disclosed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP disclosed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO disclosed