SCHEMBL8586472

SCHEMBL8586472

C[C@@]12CCC[C@H]1[C@@H]1CC(Oc3ccc(Cl)cc3)C3CCCC[C@]3(C)[C@@H]1CC2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
NR1I3 Q14994 1/20 0.37
GRIN1 Q05586 5/20 0.36
GRIN2B Q13224 5/20 0.36
SHBG P04278 1/20 0.34
STS P08842 1/20 0.34
CYP19A1 P11511 3/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MBOAT4 Q96T53 1/20 0.31
AKR1B10 O60218 1/20 0.31
LSS P48449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8586469 1.00 CDK5 (0.37) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8585044 0.87 CDK5 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8585049 0.87 CDK5 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8582194 0.85 GRIN1 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8582196 0.85 GRIN1 (0.36) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8584766 0.81 MBOAT4 (0.33) CDK5CDK5R1NR1I3SHBGSTS
SCHEMBL8584763 0.81 MBOAT4 (0.33) CDK5CDK5R1NR1I3SHBGSTS
SCHEMBL8585574 0.81 GRIN1 (0.43) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL8585577 0.81 GRIN1 (0.43) CDK5CDK5R1NR1I3GRIN1GRIN2B
SCHEMBL4728085 0.79 CDK5 (0.34) CDK5CDK5R1STSCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed