SCHEMBL8587743

SCHEMBL8587743

CCOC(=O)c1cccc2ncc(C)n12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.48
IDO1 P14902 5/20 0.45
CYP1A2 P05177 3/20 0.45
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
TGFBR1 P36897 1/20 0.42
KDM4E B2RXH2 3/20 0.42
GLA P06280 2/20 0.42
MAPK1 P28482 1/20 0.42
CYP3A4 P08684 2/20 0.41
GABRA1 P14867 2/20 0.41
GABRB2 P47870 2/20 0.41
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
LMNA P02545 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7875409 0.88 GAA (0.51) GAAIDO1CYP1A2CA12CA1
SCHEMBL12549868 0.86 CYP1A2 (0.43) GAAIDO1CYP1A2CA12CA1
SCHEMBL12549923 0.86 IDO1 (0.44) GAAIDO1CYP1A2CA12CA1
SCHEMBL7875517 0.86 GAA (0.43) GAAIDO1CYP1A2CA12CA1
SCHEMBL7868745 0.84 IDO1 (0.40) GAAIDO1CYP1A2CA12CA1
SCHEMBL7863514 0.82 IDO1 (0.42) GAAIDO1CYP1A2CA12CA1
SCHEMBL7863426 0.81 PTGS1 (0.46) GAAIDO1CYP1A2TGFBR1KDM4E
SCHEMBL7875527 0.81 GAA (0.40) GAAIDO1CYP1A2CA12CA1
Iodide SCHEMBL7868763 0.80 GAA (0.39) GAAIDO1CYP1A2CA12CA1
Trimethylammonium SCHEMBL7868762 0.80 GAA (0.39) GAAIDO1CYP1A2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998029136-A1 STABILIZED TRICYCLIC COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-07-09 WO disclosed