SCHEMBL8593107

SCHEMBL8593107

COc1ccccc1C(C)NC(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.56
CA2 P00918 5/20 0.56
ACHE P22303 2/20 0.56
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
CA12 O43570 1/20 0.48
CA4 P22748 1/20 0.48
CA14 Q9ULX7 1/20 0.48
HTR2A P28223 2/20 0.42
SLC6A4 P31645 2/20 0.42
CYP2D6 P10635 2/20 0.42
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
LPAR1 Q92633 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
ADRA2B P18089 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16179840 0.83 CA1 (0.48) CA1CA2ACHECA7CA9
SCHEMBL15473849 0.81 CYP2D6 (0.61) CA1CA2ACHECA7CA9
SCHEMBL2401390 0.81 CYP2D6 (0.61) CA1CA2ACHECA7CA9
SCHEMBL15247593 0.81 CA1 (0.58) CA1CA2ACHECA7CA9
SCHEMBL19286309 0.81 CA1 (0.58) CA1CA2ACHECA7CA9
SCHEMBL20376231 0.81 CYP2D6 (0.61) CA1CA2ACHECA7CA9
SCHEMBL24018774 0.80 KCNK3 (0.44) CA1CA2ACHEHTR2ASLC6A4
SCHEMBL22957652 0.80 KCNK3 (0.44) CA1CA2ACHEHTR2ASLC6A4
SCHEMBL20630766 0.77 CA1 (0.42) CA1CA2ACHECA7CA9
SCHEMBL22957863 0.76 CA1 (0.53) CA1CA2ACHECA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672032-B1 NOVEL PHENYLETHYL AND PHENYLPROPYLAMINES ASTRA AB (SE) 1998-01-07 EP disclosed
US-5693630-A FOR TREATMENT OF PSYCHIATRIC DISORDERS ASTRA AKTIEBOLAG (SE) 1997-12-02 US disclosed
EP-0672032-A1 NOVEL PHENYLETHYL AND PHENYLPROPYLAMINES Astra Aktiebolag (SE) 1995-09-20 EP disclosed
WO-1995009835-A1 NOVEL PHENYLETHYL AND PHENYLPROPYLAMINES ASTRA AKTIEBOLAG (SE) 1995-04-13 WO disclosed