SCHEMBL8594690

SCHEMBL8594690

CCOC(=O)NCCCN1CCCCC1C

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
TSHR P16473 1/20 0.54
HSD17B10 Q99714 2/20 0.48
SCN1A P35498 1/20 0.48
SCN2A Q99250 1/20 0.48
SCN3A Q9NY46 1/20 0.48
CXCR4 P61073 6/20 0.48
ACHE P22303 1/20 0.48
BACE1 P56817 1/20 0.48
CYP3A4 P08684 2/20 0.47
LMNA P02545 1/20 0.46
KDM4E B2RXH2 1/20 0.46
THRB P10828 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CACNA1G O43497 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8594694 1.00 CYP2D6 (0.54) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL13888624 0.81 CYP2D6 (0.56) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL2088330 0.79 HRH3 (0.57) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL19658452 0.78 CYP2D6 (0.53) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL17589298 0.77 CYP2D6 (0.50) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL17589308 0.77 CYP2D6 (0.52) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL9541617 0.76 OPRD1 (0.63) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL14156863 0.76 CXCR4 (0.54) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
Ethyl Acetate SCHEMBL11609811 0.76 SCN1A (0.48) CYP2D6CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL19718782 0.76 HRH3 (0.60) CYP2D6SCN1ASCN2ASCN3AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883613-A1 SULFONAMIDE DERIVATIVES AS 5HT7 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-12-16 EP disclosed
WO-1997029097-A1 SULFONAMIDE DERIVATIVES AS 5HT7 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-08-14 WO disclosed