SCHEMBL8598342

SCHEMBL8598342

CCc1nc2c([N+](=O)[O-])cccc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
PKN1 Q16512 1/20 0.55
PKN2 Q16513 1/20 0.55
ADORA3 P0DMS8 1/20 0.49
MGAM O43451 1/20 0.49
SI P14410 1/20 0.49
MGAM2 Q2M2H8 1/20 0.49
DDAH1 O94760 1/20 0.46
PDE10A Q9Y233 1/20 0.44
NOS1 P29475 3/20 0.42
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
NOS2 P35228 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1892570 0.88 KDM4E (0.52) GAAPKN1PKN2ADORA3MGAM
SCHEMBL6995989 0.88 PKN1 (0.57) GAAPKN1PKN2ADORA3MGAM
SCHEMBL7486947 0.85 PKN1 (0.52) GAAPKN1PKN2ADORA3MGAM
SCHEMBL15228495 0.85 PKN1 (0.55) GAAPKN1PKN2ADORA3MGAM
SCHEMBL4888425 0.85 PKN1 (0.55) GAAPKN1PKN2ADORA3MGAM
SCHEMBL3947018 0.85 PKN1 (0.55) GAAPKN1PKN2ADORA3MGAM
SCHEMBL8328888 0.84 PKN1 (0.51) GAAPKN1PKN2ADORA3MGAM
SCHEMBL7475180 0.84 PKN1 (0.51) GAAPKN1PKN2ADORA3MGAM
Hydrochloric Acid SCHEMBL4882337 0.84 PKN1 (0.53) GAAPKN1PKN2ADORA3MGAM
SCHEMBL7479338 0.82 PKN1 (0.52) GAAPKN1PKN2ADORA3MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017064675-A1 HINDERED DISULFIDE DRUG CONJUGATES GENENTECH, INC. (US) 2017-04-20 WO disclosed
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed