SCHEMBL8599595

SCHEMBL8599595

Cc1cccc(C)c1C(=O)Nc1cccc2c1nc(C(F)(F)F)n2CC(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
ALDH1A1 P00352 2/20 0.39
APEX1 P27695 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDR P35968 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 3/20 0.37
GAA P10253 1/20 0.37
CYP3A4 P08684 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8600640 0.92 TP53 (0.53) TP53CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8597312 0.87 TP53 (0.43) TP53CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8601785 0.87 TP53 (0.48) TP53CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8602071 0.84 MAPT (0.46) TP53ALDH1A1KDM4ESMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL8601062 0.80 TP53 (0.47) TP53ALDH1A1KDM4EHTTKMT2A
SCHEMBL8596165 0.80 TP53 (0.45) TP53CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8601684 0.78 RXFP1 (0.44) TP53ALDH1A1APEX1KDM4EHPGD
SCHEMBL8598838 0.78 TP53 (0.43) TP53CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8597937 0.78 TP53 (0.43) TP53SMN1; SMN2HTTMEN1KMT2A
Trifluoroacetic Acid SCHEMBL8598750 0.76 CDK4 (0.42) ALDH1A1SMN1; SMN2HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed