SCHEMBL8599778

SCHEMBL8599778

O=CCC1Cc2cc(F)c(F)cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.37
METAP1 P53582 6/20 0.37
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873406 1.00 ACHE (0.37) ACHEMETAP1CYP2C9KCNH2
SCHEMBL8595469 0.83 ACHE (0.38) ACHEMETAP1CYP2C9KCNH2
SCHEMBL8595473 0.83 ACHE (0.38) ACHEMETAP1CYP2C9KCNH2
SCHEMBL8874743 0.83 ACHE (0.38) ACHEMETAP1CYP2C9KCNH2
SCHEMBL8873213 0.81 METAP1 (0.43) ACHEMETAP1
SCHEMBL8598434 0.81 METAP1 (0.43) ACHEMETAP1
SCHEMBL8873958 0.81 ACHE (0.55) ACHEMETAP1
SCHEMBL8873012 0.81 DRD3 (0.49) ACHEMETAP1
SCHEMBL8599815 0.81 DRD3 (0.49) ACHEMETAP1
SCHEMBL8594761 0.81 ACHE (0.55) ACHEMETAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed