SCHEMBL8600057

SCHEMBL8600057

COc1cc(COc2cc(N)c(Cl)cc2C(CCCC=O)N2CCC(C)CC2)cc(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
ACHE P22303 1/20 0.33
ENPP2 Q13822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603836 0.92 MEN1 (0.40) MEN1ALDH1A1TP53CYP3A4CYP2D6
SCHEMBL8601233 0.92 MEN1 (0.39) MEN1ALDH1A1TP53CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8599772 0.92 MEN1 (0.39) MEN1ALDH1A1TP53CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8599756 0.92 MEN1 (0.40) MEN1ALDH1A1TP53CYP3A4CYP2D6
SCHEMBL8602358 0.91 CYP3A4 (0.38) MEN1ALDH1A1TP53CYP3A4CYP2D6
SCHEMBL8600560 0.90 MEN1 (0.44) MEN1ALDH1A1TP53CYP3A4CYP2D6
SCHEMBL8601824 0.90 KMT2A (0.41) MEN1ALDH1A1TP53CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8599724 0.90 KMT2A (0.40) MEN1ALDH1A1TP53CYP3A4CYP2D6
SCHEMBL8604410 0.89 MEN1 (0.37) MEN1ALDH1A1TP53CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8603573 0.89 MEN1 (0.44) MEN1ALDH1A1TP53CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed