SCHEMBL8600182

SCHEMBL8600182

Cc1cn(Cc2ccc3c(c2)OCO3)c2cc(CC(=O)O)ccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 9/20 0.76
PDE4A P27815 1/20 0.59
PDE4B Q07343 1/20 0.59
PDE4C Q08493 1/20 0.59
PDE4D Q08499 1/20 0.59
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA7 P36544 1/20 0.47
CHRNA4 P43681 1/20 0.47
RAB9A P51151 1/20 0.45
MAPK10 P53779 1/20 0.44
HIF1A Q16665 1/20 0.44
EDNRB P24530 1/20 0.44
EDNRA P25101 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1553375 0.87 PDE4A (0.67) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL11977182 0.86 SLC22A12 (1.00) SLC22A12PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL8601429 0.86 PDE4A (0.66) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL8601425 0.83 PDE4A (0.69) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL1554280 0.82 PDE4A (0.64) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL8602152 0.81 SLC22A12 (0.78) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL8604805 0.80 SLC22A12 (0.74) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL8572873 0.79 SLC22A12 (0.70) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL3944098 0.78 CYP3A4 (0.75) ALDH1A1CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL29642680 0.78 CYP3A4 (0.75) ALDH1A1CYP1A2CYP3A4CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed