SCHEMBL8600387

SCHEMBL8600387

C=C(C(=O)OC)c1ccc2nc[nH]c2c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.58
RAB9A P51151 5/20 0.56
NPC1 O15118 5/20 0.56
KMT2A Q03164 4/20 0.56
SMN1; SMN2 Q16637 4/20 0.54
HTT P42858 3/20 0.54
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 1/20 0.54
HPGD P15428 1/20 0.54
POLB P06746 7/20 0.52
TDP1 Q9NUW8 3/20 0.51
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
CTNNB1 P35222 1/20 0.50
WNT3A P56704 1/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.49
MMP12 P39900 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8600378 0.89 HDAC6 (0.44) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL1379300 0.82 KMT2A (0.65) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL29465824 0.82 KMT2A (0.65) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL5542915 0.81 KMT2A (0.64) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL5131245 0.81 HDAC6 (0.59) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
Sulfuric Acid SCHEMBL7332404 0.77 KMT2A (0.60) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL3776194 0.77 HDAC6 (0.66) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL5777206 0.77 HDAC6 (0.66) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL11172 0.76 HDAC6 (0.74) HDAC6RAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL30265442 0.76 HDAC6 (0.74) HDAC6RAB9ANPC1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871624-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE Merck & Co., Inc. (US) 1998-10-21 EP disclosed
WO-1997021703-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO., INC. (US) 1997-06-19 WO disclosed