SCHEMBL8600489

SCHEMBL8600489

c1csc(C2COCCN2)n1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BAZ2A Q9UIF9 1/20 0.37
CSNK1D P48730 1/20 0.34
CSNK1E P49674 1/20 0.34
KCNH2 Q12809 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.33
HTR2C P28335 1/20 0.33
PRKACA P17612 1/20 0.31
PRKACG P22612 1/20 0.31
PRKACB P22694 1/20 0.31
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL551606 0.75 CHRNB2 (0.43)
SCHEMBL7750646 0.74
SCHEMBL18903009 0.74
Hydrochloric Acid SCHEMBL19259428 0.74 CHRNB2 (0.42) HTR2C
SCHEMBL978739 0.74 MEN1 (0.45) BAZ2AHTR2C
SCHEMBL29285276 0.72 DRD3 (0.36) HTR2CNOS3NOS2
SCHEMBL787918 0.72 CHRM2 (0.39) HTR2CNOS3NOS2
SCHEMBL24540766 0.72 CSNK1D (0.36) BAZ2ACSNK1DCSNK1EKCNH2PRKACA
Hydrochloric Acid SCHEMBL4573925 0.71 CHRM2 (0.38) HTR2CNOS3NOS2
SCHEMBL31610616 0.70 PIK3C3 (0.35) PIK3C3NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110431138-A AR-V7 inhibitor HOFFMANN LA ROCHE 2019-11-08 CN claimed
CN-110431138-A AR-V7 inhibitor HOFFMANN LA ROCHE 2019-11-08 CN disclosed
CN-106164071-B Human androgenic receptor DNA- binding structural domain (DBD) compound and its application method as therapeutic agent 不列颠哥伦比亚大学 2019-09-10 CN disclosed
EP-0345593-B2 2-substituted coumaran derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-02-04 EP disclosed
EP-0345593-A1 2-substituted coumaran derivatives Takeda Chemical Industries, Ltd. (JP) 1989-12-13 EP disclosed