SCHEMBL8600788

SCHEMBL8600788

CC(=O)Oc1c(C)cc(OC=C(C)C)c(C)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
POLB P06746 1/20 0.45
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 3/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
ACHE P22303 3/20 0.35
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910532 0.82 POLB (0.62) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL13954030 0.79 POLB (0.54) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL4495765 0.78 HTT (0.43) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL4495767 0.78 HTT (0.43) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL14407309 0.77 HTT (0.59) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL4492895 0.76 HTT (0.44) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL10941837 0.76 KDM4E (0.49) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL10624847 0.76 KDM4E (0.52) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL9596191 0.74 HTT (0.47) HTTPOLBKDM4EHSD17B10GAA
SCHEMBL8600805 0.73 HTT (0.44) HTTPOLBKDM4EHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345593-B2 2-substituted coumaran derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-02-04 EP disclosed
EP-0345592-B1 NOVEL 2-SUBSTITUTED COUMARAN DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1993-08-11 EP disclosed
US-4978761-A Enzyme inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-12-18 US disclosed
US-4966973-A LIPOXYGENASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-10-30 US disclosed
EP-0345593-A1 2-substituted coumaran derivatives Takeda Chemical Industries, Ltd. (JP) 1989-12-13 EP disclosed
EP-0345592-A1 Novel 2-substituted coumaran derivatives Takeda Chemical Industries, Ltd. (JP) 1989-12-13 EP disclosed