SCHEMBL8601355

SCHEMBL8601355

CNc1nc2c([N+](=O)[O-])cccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.55
PKN2 Q16513 1/20 0.55
ADORA3 P0DMS8 1/20 0.49
MGAM O43451 1/20 0.49
GAA P10253 1/20 0.49
SI P14410 1/20 0.49
MGAM2 Q2M2H8 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.45
RAB9A P51151 2/20 0.45
NPC1 O15118 2/20 0.44
PDE10A Q9Y233 1/20 0.44
NOS1 P29475 4/20 0.42
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 3/20 0.41
NOS2 P35228 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7954749 0.85 PKN1 (0.49) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7954751 0.85 PKN1 (0.49) PKN1PKN2ADORA3MGAMGAA
Dimethylamine SCHEMBL7486960 0.83 PKN1 (0.56) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7486053 0.83 PKN1 (0.50) PKN1PKN2ADORA3MGAMGAA
SCHEMBL1013853 0.83 LMNA (0.54) PKN1PKN2ADORA3MGAMGAA
SCHEMBL6332531 0.82 PKN1 (0.61) PKN1PKN2ADORA3MGAMGAA
SCHEMBL8328888 0.81 PKN1 (0.51) PKN1PKN2ADORA3MGAMGAA
SCHEMBL1013588 0.81 PKN1 (0.60) PKN1PKN2ADORA3MGAMGAA
SCHEMBL11020624 0.79 PKN1 (0.49) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7016736 0.79 PKN1 (0.46) PKN1PKN2ADORA3MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed