SCHEMBL8601975

SCHEMBL8601975

Fc1cccnc1C1CCCCN1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.51
CHRNA4 P43681 3/20 0.51
MEN1 O00255 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C19 P33261 2/20 0.51
KMT2A Q03164 2/20 0.51
CHRNA7 P36544 2/20 0.51
POLB P06746 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2A6 P11509 1/20 0.51
CYP2C9 P11712 1/20 0.51
AURKA O14965 1/20 0.44
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRM5 P08912 2/20 0.36
CHRM3 P20309 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23178137 0.95 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL28485125 0.95 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL30582955 0.95 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL21516009 0.81 CHRNB2 (0.51) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL15237647 0.81 CHRNB2 (0.51) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL6131954 0.77 CXCR4 (0.36) HTR1ASLC6A2SLC6A4
SCHEMBL21516103 0.75 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL31444389 0.75 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL20851551 0.75 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19
SCHEMBL24694986 0.75 CHRNB2 (0.50) CHRNB2CHRNA4MEN1CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719166-A TREATING PSYCHOSES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1998-02-17 US disclosed
EP-0532177-B1 Methanoanthracenes as dopamine antagonists ZENECA LTD (GB) 1996-10-16 EP disclosed
US-5550136-A ANTAGONISTS OF DOPAMINE D-2 RECEPTORS ZENECA LIMITED (GB) 1996-08-27 US disclosed
US-5399568-A Dopamine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-21 US disclosed
EP-0532177-A1 Methanoanthracenes as dopamine antagonists ZENECA LIMITED (GB) 1993-03-17 EP disclosed