SCHEMBL8604236

SCHEMBL8604236

CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CC(=O)N3)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 8/20 0.58
RARG P13631 7/20 0.58
RARA P10276 6/20 0.47
CYP3A4 P08684 2/20 0.47
KMT2A Q03164 1/20 0.47
HDAC3 O15379 6/20 0.43
HDAC4 P56524 6/20 0.43
HDAC1 Q13547 6/20 0.43
HDAC2 Q92769 6/20 0.43
HDAC8 Q9BY41 6/20 0.43
HDAC6 Q9UBN7 6/20 0.43
HDAC9 Q9UKV0 6/20 0.43
CYP26A1 O43174 1/20 0.42
CRABP2 P29373 1/20 0.42
MAPK1 P28482 1/20 0.41
AKR1B1 P15121 1/20 0.41
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
MDH2 P40926 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8866305 0.91 RARB (0.71) RARBRARGRARACYP3A4KMT2A
SCHEMBL8606002 0.88 RARB (0.47) RARBRARGRARACYP3A4KMT2A
SCHEMBL8867050 0.83 RARB (0.81) RARBRARGRARACYP3A4HDAC3
SCHEMBL8565867 0.82 RARB (0.71) RARBRARGRARACYP3A4KMT2A
SCHEMBL8606006 0.81 RARB (0.46) RARBRARGRARACYP3A4KMT2A
SCHEMBL9023692 0.79 RARB (0.48) RARBRARGRARACYP3A4KMT2A
SCHEMBL8631973 0.79 RARB (0.55) RARBRARGRARACYP3A4KMT2A
SCHEMBL9484975 0.79 RARB (0.67) RARBRARGRARACYP3A4KMT2A
SCHEMBL8634168 0.76 RARB (0.74) RARBRARGRARACYP3A4KMT2A
SCHEMBL5737002 0.76 RARB (0.52) RARBRARGRARACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP disclosed
US-5616712-A SKIN DISORDERS; ANTICARCINOGENIC AND -INFLAMMATORY AGENTS; AUTOIMMUNE DISEASES; ALLERGAN (US) 1997-04-01 US disclosed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO disclosed