SCHEMBL8565867

SCHEMBL8565867

CCOC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CCN3)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 12/20 0.71
RARG P13631 9/20 0.71
RARA P10276 9/20 0.71
CYP3A4 P08684 4/20 0.52
KMT2A Q03164 1/20 0.52
CYP26A1 O43174 2/20 0.47
CRABP2 P29373 1/20 0.47
HSPA9 P38646 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ESR1 P03372 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
ESR2 Q92731 1/20 0.39
CA14 Q9ULX7 1/20 0.39
MMP13 P45452 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1485938 0.88 RARB (0.69) RARBRARGRARACYP3A4KMT2A
SCHEMBL9484975 0.83 RARB (0.67) RARBRARGRARACYP3A4KMT2A
SCHEMBL8604236 0.82 RARB (0.58) RARBRARGRARACYP3A4KMT2A
SCHEMBL8671725 0.82 RARB (0.53) RARBRARGRARACYP3A4KMT2A
SCHEMBL8606002 0.81 RARB (0.47) RARBRARGRARACYP3A4KMT2A
SCHEMBL8606006 0.81 RARB (0.46) RARBRARGRARACYP3A4KMT2A
SCHEMBL10693400 0.80 RARB (0.53) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10693407 0.80 RARB (0.53) RARBRARGRARACYP3A4CYP26A1
SCHEMBL444860 0.79 RARB (0.78) RARBRARGRARACYP3A4KMT2A
SCHEMBL9056981 0.78 ALDH1A1 (0.47) RARBRARGRARAKMT2AHSPA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5717094-A 6-THIOCHROMANYL-ETHYNE, 6-CHROMANYL ETHYNE AND 6-TETRAHYDROQUINOLINYL ETHYNE OR THEIR METAL SALTS ARE REACTED WITH SUITABLE HALO SUBSTITUTED PHENYL OR HETEROARYL COMPUNDS ALLERGAN (US) 1998-02-10 US disclosed
CN-1028174-C Process and intermediates for preparing compounds having disubstituted acetylene moiety and retinoic acid-like biological activity ALLERGAN INC (US) 1995-04-12 CN disclosed
CN-1050385-A Preparation has bioactive method and the intermediate that has the compound of disubstituted acetylene moiety of retinoic acid-like ALLERGAN INC (US) 1991-04-03 CN disclosed