SCHEMBL8607463

SCHEMBL8607463

O=C(O)c1cn2cccc(CCC(O)c3nnn[nH]3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
RXFP1 Q9HBX9 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
DHODH Q02127 1/20 0.31
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8607749 0.89 PTGS1 (0.39) PTGS1PTGS2RXFP1HTR2AHTR2C
SCHEMBL8608469 0.86 PTGS1 (0.34) PTGS1PTGS2RXFP1CREBBP
SCHEMBL8606176 0.82 PTGS1 (0.40) PTGS1PTGS2RXFP1HTR2AHTR2C
SCHEMBL8609477 0.82 KDM4E (0.30)
SCHEMBL8605302 0.81 PTGS1 (0.39) PTGS1PTGS2RXFP1HTR2AHTR2C
SCHEMBL8609715 0.79 PTGS1 (0.36) PTGS1PTGS2RXFP1DHODHCREBBP
SCHEMBL9753569 0.78 PTGS1 (0.39) PTGS1PTGS2
SCHEMBL8607312 0.78 RXFP1 (0.32) PTGS1PTGS2RXFP1
SCHEMBL2505187 0.72 PTGS1 (0.51) PTGS1PTGS2RXFP1DHODHCREBBP
SCHEMBL8606992 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716964-A BRAIN DISORDERS; ANTIISCHEMIC AGENTS G.D. SEARLE & CO. (US) 1998-02-10 US disclosed