SCHEMBL8609211

SCHEMBL8609211

O=C(O)c1cn2cc(CP(=O)(O)O)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
EGLN1 Q9GZT9 11/20 0.46
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
METTL3 Q86U44 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25308496 0.81 EGLN1 (0.46) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL8607604 0.80 PTGS1 (0.50) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL3498034 0.78 PTGS1 (0.58) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL8607242 0.78 P4HTM (0.50) PTGS1PTGS2EGLN1
SCHEMBL8608756 0.77 PTGS1 (0.53) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL8608817 0.75 TBXAS1 (0.49) PTGS1PTGS2EGLN1CYP1A2MAPT
SCHEMBL8346854 0.75 PTGS1 (0.35) PTGS1PTGS2CYP1A2CYP3A4MAPT
SCHEMBL8609927 0.75 PTGS1 (0.48) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL8609437 0.73 PTGS1 (0.46) PTGS1PTGS2EGLN1CYP1A2CYP3A4
SCHEMBL28626437 0.73 PTGS1 (0.59) PTGS1PTGS2EGLN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633237-A Imidazo[1,2-a]pyridinylalkyl phosphonic acid compounds for treatment of neurotoxic injury G.D. SEARLE & CO. (US) 1997-05-27 US claimed
US-5360796-A Treatment of hypoxia, anoxia or ischemia G. D. SEARLE & CO. (US) 1994-11-01 US claimed
EP-0436831-A2 Imidazo[1,2-a]pyridinylalkyl compounds for treatment of neurotoxic injury G.D. Searle & Co. (US) 1991-07-17 EP claimed
WO-1991008211-A1 IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF NEUROTOXIC INJURY G.D. SEARLE & CO. (US) 1991-06-13 WO claimed
US-5716964-A BRAIN DISORDERS; ANTIISCHEMIC AGENTS G.D. SEARLE & CO. (US) 1998-02-10 US disclosed
US-5633237-A Imidazo[1,2-a]pyridinylalkyl phosphonic acid compounds for treatment of neurotoxic injury G.D. SEARLE & CO. (US) 1997-05-27 US disclosed
US-5360796-A Treatment of hypoxia, anoxia or ischemia G. D. SEARLE & CO. (US) 1994-11-01 US disclosed
EP-0436831-A2 Imidazo[1,2-a]pyridinylalkyl compounds for treatment of neurotoxic injury G.D. Searle & Co. (US) 1991-07-17 EP disclosed
WO-1991008211-A1 IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF NEUROTOXIC INJURY G.D. SEARLE & CO. (US) 1991-06-13 WO disclosed