SCHEMBL8610247

SCHEMBL8610247

O[C@H]1[C@@H](OC(c2ccccc2)(c2ccccc2)c2ccccc2)[C@H](n2cnc3cncnc32)O[C@@H]1COC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYMP P19971 14/20 0.57
ADORA1 P30542 2/20 0.47
DNMT3B Q9UBC3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613308 0.93 TYMP (0.57) TYMPADORA1DNMT3B
SCHEMBL8610677 0.91 TYMP (0.68) TYMPADORA1DNMT3B
SCHEMBL8610715 0.87 TYMP (0.48) TYMPADORA1DNMT3B
SCHEMBL8610717 0.87 TYMP (0.48) TYMPADORA1DNMT3B
SCHEMBL8613137 0.85 TYMP (0.51) TYMPADORA1
SCHEMBL8612903 0.85 TYMP (0.51) TYMPADORA1
SCHEMBL8611837 0.83 TYMP (0.67) TYMPADORA1
SCHEMBL8613000 0.83 TYMP (0.83) TYMPADORA1
SCHEMBL31438688 0.82 TYMP (0.52) TYMPADORA1DNMT3B
SCHEMBL21427352 0.82 TYMP (0.56) TYMPADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO claimed
US-5750675-A 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosylpurines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1998-05-12 US disclosed
US-5525720-A Synthesis of 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosyl purines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1996-06-11 US disclosed
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO disclosed