SCHEMBL8610346

SCHEMBL8610346

CCCOc1ccccc1C(C)(C)C.C[Si](C)(C)C#CCO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 4/20 0.46
GAA P10253 4/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
NPSR1 Q6W5P4 3/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
MAPK1 P28482 1/20 0.38
MAPT P10636 3/20 0.38
NISCH Q9Y2I1 1/20 0.38
P2RY1 P47900 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8609507 0.91 ALDH1A1 (0.52) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL8609250 0.83 ALDH1A1 (0.38) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL8610692 0.83 ALDH1A1 (0.52) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL10603372 0.81 CYP1A2 (0.58) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL8610693 0.74 ALDH1A1 (0.59) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL10787315 0.73 ALDH1A1 (0.58) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL8142983 0.73 ALDH1A1 (0.65) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL11133824 0.72 ALDH1A1 (0.60) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL23007678 0.70 CYP1A2 (0.45) ALDH1A1KDM4EGAACYP1A2CYP2D6
SCHEMBL9515076 0.69 ALDH1A1 (0.55) ALDH1A1KDM4EGAACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP disclosed
EP-0661258-A1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1995-07-05 EP disclosed