SCHEMBL8611432

SCHEMBL8611432

Cc1cccc(NC(=O)N[C@H]2N=C(c3ccccc3)c3ccccc3NC2=S)c1

nearest known ligand 0.82

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 11/20 0.82
KCNH2 Q12809 1/20 0.63
CCKAR P32238 3/20 0.58
CYP3A4 P08684 1/20 0.57
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9468540 1.00 CCKBR (0.82) CCKBRKCNH2CCKARCYP3A4MAPT
SCHEMBL8681438 1.00 CCKBR (0.82) CCKBRKCNH2CCKARCYP3A4MAPT
SCHEMBL641958 0.90 CCKBR (1.00) CCKBRKCNH2CCKARCYP3A4MAPT
SCHEMBL8682548 0.88 CCKBR (0.64) CCKBRKCNH2CCKAR
SCHEMBL9865815 0.87 CCKBR (0.65) CCKBRKCNH2
SCHEMBL9468952 0.82 CCKBR (0.81) CCKBR
SCHEMBL8681481 0.82 CCKBR (0.81) CCKBR
SCHEMBL9109762 0.82 CCKBR (0.64) CCKBRCCKAR
SCHEMBL642143 0.82 CCKBR (0.85) CCKBRCCKAR
SCHEMBL8681334 0.80 CCKBR (0.63) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730456-A4 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO INC (US) 1998-02-04 EP disclosed
EP-0730456-A1 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO. INC. (US) 1996-09-11 EP disclosed
WO-1995014472-A1 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO., INC. (US) 1995-06-01 WO disclosed