SCHEMBL8611564

SCHEMBL8611564

Nc1cc(Cl)c(-n2cccc2)cc1N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.46
KDM4E B2RXH2 2/20 0.46
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 3/20 0.41
PKM P14618 1/20 0.41
CD44 P16070 1/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
LMNA P02545 2/20 0.36
MAPT P10636 3/20 0.34
CYP3A4 P08684 3/20 0.34
NFKB1 P19838 1/20 0.34
PMP22 Q01453 1/20 0.34
TSHR P16473 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIA1 P42261 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA3 P42263 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640129 0.89 GAA (0.52) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL11830148 0.82 GAA (0.46) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL30758081 0.82 GAA (0.46) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL8296289 0.79 CA12 (0.36) GAAKDM4EPOLBALDH1A1CD44
SCHEMBL10914973 0.74 KDM4E (0.50) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL10913318 0.74 CYP3A4 (0.56) GAAKDM4EPOLBALDH1A1PKM
SCHEMBL29266693 0.73 POLB (0.42) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL8977414 0.73 KDM4E (0.46) GAAKDM4EALDH1A1PKMLMNA
SCHEMBL13480887 0.71 POLB (0.45) GAAKDM4EPOLBL3MBTL1ALDH1A1
SCHEMBL22636601 0.71 AHR (0.42) GAAKDM4EPOLBL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852017-A 2,3(1H,4H)-quinoxalinediones BASF AKTIENGESELLSCHAFT (DE) 1998-12-22 US disclosed
EP-0572852-B1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF AG (DE) 1998-10-21 EP disclosed
US-5714489-A 2,3(1H,4H)quinoxalinedione BASF AKTIENGESELLSCHAFT (DE) 1998-02-03 US disclosed
EP-0572852-A1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF Aktiengesellschaft (DE) 1993-12-08 EP disclosed