SCHEMBL8612671

SCHEMBL8612671

CC(=O)Nc1ccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.65
MEN1 O00255 6/20 0.65
KDM4E B2RXH2 4/20 0.57
PDE10A Q9Y233 2/20 0.57
ALDH1A1 P00352 7/20 0.54
CYP1A2 P05177 2/20 0.54
TP53 P04637 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CYP3A4 P08684 4/20 0.54
MOK Q9UQ07 3/20 0.53
KCNH2 Q12809 2/20 0.53
HPGD P15428 2/20 0.53
TACR3 P29371 1/20 0.53
ALOX12 P18054 2/20 0.52
CYP2C19 P33261 1/20 0.52
MAPT P10636 3/20 0.51
POLB P06746 1/20 0.51
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617762 0.93 KMT2A (0.64) KMT2AMEN1KDM4EPDE10AALDH1A1
SCHEMBL8619408 0.89 MEN1 (0.51) KMT2AMEN1KDM4EALDH1A1CYP1A2
SCHEMBL8613680 0.87 ALDH1A1 (0.48) KMT2AMEN1KDM4EPDE10AALDH1A1
SCHEMBL8615144 0.85 CA9 (0.51) KMT2AMEN1KDM4EALDH1A1CYP1A2
SCHEMBL8613473 0.85 ADORA1 (0.51) KMT2AMEN1KDM4EALDH1A1CYP1A2
SCHEMBL8617733 0.84 CYP3A4 (0.58) KMT2AMEN1KDM4EPDE10AALDH1A1
SCHEMBL8617743 0.84 CYP3A4 (0.65) KMT2AMEN1KDM4EPDE10AALDH1A1
SCHEMBL8615206 0.83 CYP3A4 (0.52) KMT2AMEN1KDM4EPDE10AALDH1A1
SCHEMBL8615933 0.83 CYP3A4 (0.52) KMT2AMEN1KDM4EPDE10AALDH1A1
Hydrochloric Acid SCHEMBL8620745 0.83 CYP3A4 (0.64) KMT2AMEN1KDM4EPDE10AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed