SCHEMBL8613632

SCHEMBL8613632

O=CNNC1CCCc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
EPHX1 P07099 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.49
TAS1R3 Q7RTX0 3/20 0.48
TAS1R1 Q7RTX1 3/20 0.48
CYP1A2 P05177 1/20 0.48
TAS1R2 Q8TE23 2/20 0.48
KDM4E B2RXH2 1/20 0.47
CYP2D6 P10635 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28265320 0.90 PDPK1 (0.56) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL2115700 0.84 HTT (0.63) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL3532080 0.83 HTT (0.55) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL3532081 0.83 HTT (0.55) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL6001031 0.83 HTT (0.55) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL24106055 0.82 EPHX1 (0.51) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL11748233 0.81 HTT (0.60) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL6810979 0.79 EPHX1 (0.62) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL27480299 0.78 PDPK1 (0.58) HTTKMT2AMEN1EPHX1SMN1; SMN2
SCHEMBL22525050 0.76 ALDH1A1 (0.54) HTTKMT2AMEN1EPHX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed