SCHEMBL8613823

SCHEMBL8613823

CC(C)(C)S(=O)(=O)Nc1ccc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 7/20 0.48
CA12 O43570 4/20 0.48
CA1 P00915 4/20 0.48
CA2 P00918 4/20 0.48
MAPT P10636 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
CYP3A4 P08684 4/20 0.45
TACR3 P29371 1/20 0.45
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 4/20 0.44
HPGD P15428 1/20 0.44
KCNH2 Q12809 1/20 0.44
CNR1 P21554 2/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613739 0.89 ALDH1A1 (0.51) CA9CA12CA1CA2MAPT
SCHEMBL8616347 0.87 ALDH1A1 (0.53) CA9CA12CA1CA2MAPT
SCHEMBL8613821 0.84 CA9 (0.46) CA9CA12CA1CA2MAPT
SCHEMBL8613671 0.83 TACR3 (0.53) CA9CA12CA1CA2MAPT
SCHEMBL8617762 0.83 KMT2A (0.64) CA9CA12CA1CA2MAPT
SCHEMBL8613501 0.82 CA9 (0.45) CA9CA12CA1CA2MAPT
SCHEMBL8615144 0.82 CA9 (0.51) CA9CA12CA1CA2MAPT
SCHEMBL8616004 0.81 KDM4E (0.61) CA9CA12CA1CA2MAPT
SCHEMBL8617924 0.80 TACR3 (0.49) CA9CA12CA1CA2MAPT
SCHEMBL8613846 0.80 KDM4E (0.67) MAPTCYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed