SCHEMBL8613993

SCHEMBL8613993

Cc1c(C)c2c(c(C)c1O)CCC(C)OC(=O)CCCCO2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA9 Q16790 2/20 0.42
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
CAPN1 P07384 1/20 0.31
ALOX5 P09917 1/20 0.31
HPGD P15428 1/20 0.30
VCP P55072 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612197 0.84 CYP1A2 (0.34) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL8610857 0.81 PTGS1 (0.40) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL31314432 0.77 ALOX5 (0.41) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL1567962 0.77 ALOX5 (0.41) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL13309507 0.77 ALOX5 (0.41) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL11750965 0.77 ALOX5 (0.41) CA1CA9PTGS1PTGS2CYP1A2
Hydrochloric Acid SCHEMBL30892599 0.76 ALOX5 (0.40) CA1CA9PTGS1PTGS2CYP1A2
SCHEMBL10458358 0.74 CA1 (0.67) CA1CA9CYP1A2TSHR
SCHEMBL12713304 0.74 CYP3A4 (0.42) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL7155377 0.71 CA1 (0.59) CA1CA9CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0718295-B1 Lactones with antioxidising and hypolipidaemic activity useful in the therapy of the atherosclerosis ALFA WASSERMANN SPA (IT) 1998-04-22 EP claimed
US-5608084-A AND VASCULAR PATHOLOGIES; MULTISTEP PREPARATION BY REACTING A HYDROQUINONE WITH ALKYL VINYL KETONE, ESTERIFYING HYDROXY 3,4-DIHYDRO-2H-1-BENZOPYRAN, DEMETHYLATING ETHER, REACTING WITH ALKYL 5-BROMOPENTANOATE, HYDROLYZING, TWO MORE STEPS ALFA WASSERMANN S.P.A. (IT) 1997-03-04 US claimed
EP-0718295-A1 Lactones with antioxidising and hypolipidaemic activity useful in the therapy of the atherosclerosis ALFA WASSERMANN S.p.A. (IT) 1996-06-26 EP claimed
EP-0718295-B1 Lactones with antioxidising and hypolipidaemic activity useful in the therapy of the atherosclerosis ALFA WASSERMANN SPA (IT) 1998-04-22 EP disclosed
EP-0718295-A1 Lactones with antioxidising and hypolipidaemic activity useful in the therapy of the atherosclerosis ALFA WASSERMANN S.p.A. (IT) 1996-06-26 EP disclosed