SCHEMBL8614155

SCHEMBL8614155

CCCn1c(=O)cnc(=O)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
PGR P06401 2/20 0.48
KDM4E B2RXH2 6/20 0.47
LMNA P02545 5/20 0.47
POLB P06746 4/20 0.47
HPGD P15428 4/20 0.47
HSD17B10 Q99714 2/20 0.47
GAA P10253 1/20 0.47
TSHR P16473 3/20 0.47
MAPK1 P28482 3/20 0.47
MAPT P10636 2/20 0.47
ALOX15 P16050 2/20 0.47
USP2 O75604 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
RORA P35398 1/20 0.45
RORC P51449 1/20 0.45
RORB Q92753 1/20 0.45
ADORA3 P0DMS8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7290888 0.87 ALDH1A1 (0.61) ALDH1A1PGRKDM4ELMNAHPGD
SCHEMBL30343301 0.81 KDM4E (0.63) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL11455551 0.81 KDM4E (0.63) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL7290881 0.81 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL5995444 0.78 KDM4E (0.53) ALDH1A1PGRKDM4EPOLBHPGD
SCHEMBL13386557 0.78 ALDH1A1 (0.71) ALDH1A1PGRKDM4ELMNAPOLB
SCHEMBL28973475 0.74 KDM4E (0.68) ALDH1A1PGRKDM4ELMNAPOLB
SCHEMBL9393950 0.74 POLB (0.45) ALDH1A1KDM4EPOLBHSD17B10GAA
SCHEMBL153959 0.73 ALDH1A1 (0.62) ALDH1A1PGRKDM4ELMNAPOLB
SCHEMBL30012682 0.73 ALDH1A1 (0.62) ALDH1A1PGRKDM4ELMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730453-A4 METHODS OF TREATING CARDIAC ARRHYTHMIA MERCK & CO INC (US) 1998-03-04 EP disclosed
US-5597818-A CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1997-01-28 US disclosed
EP-0730453-A1 METHODS OF TREATING CARDIAC ARRHYTHMIA MERCK & CO. INC. (US) 1996-09-11 EP disclosed
US-5438055-A Antiarrhythmic benzodiazepines MERCK & CO., INC. (US) 1995-08-01 US disclosed
US-5428031-A Benzodiazepine analogs; cardiovascular disorders MERCK & CO., INC. (US) 1995-06-27 US disclosed
WO-1995014470-A1 METHODS OF TREATING CARDIAC ARRHYTHMIA MERCK & CO., INC. (US) 1995-06-01 WO disclosed
WO-1995014473-A1 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO., INC. (US) 1995-06-01 WO disclosed