SCHEMBL8615217

SCHEMBL8615217

CCCC(C)(C)c1cccc(-c2cc(C(=O)NC(=N)N)c3ccccc3n2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 9/20 0.53
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
LMNA P02545 2/20 0.52
HTT P42858 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 1/20 0.52
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
TACR2 P21452 2/20 0.46
PTGER4 P35408 1/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KCNH2 Q12809 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619048 0.89 TACR3 (0.47) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8617836 0.86 KDM4E (0.58) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8619426 0.85 TACR3 (0.55) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8617534 0.84 CA12 (0.64) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8617116 0.82 ALDH1A1 (0.56) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8617743 0.81 CYP3A4 (0.65) TACR3KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL8618943 0.81 MEN1 (0.65) TACR3KDM4EALDH1A1LMNAHTT
SCHEMBL8617924 0.81 TACR3 (0.49) TACR3KDM4EALDH1A1HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL8620745 0.80 CYP3A4 (0.64) TACR3KDM4EALDH1A1LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL8613665 0.80 MEN1 (0.64) TACR3KDM4EALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed