SCHEMBL8615374

SCHEMBL8615374

C[Si](C)(C)C#Cc1ccc2cccnc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
MEN1 O00255 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
KMT2A Q03164 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.47
NR4A2 P43354 1/20 0.47
PDGFRB P09619 1/20 0.45
PDGFRA P16234 1/20 0.45
GRM5 P41594 1/20 0.39
KCNH2 Q12809 1/20 0.39
CYP3A4 P08684 2/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
PDE10A Q9Y233 1/20 0.37
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30600696 0.87 ALDH1A1 (0.51) ALDH1A1MEN1CASP1KMT2AHTT
SCHEMBL6852232 0.79 ALDH1A1 (0.50) ALDH1A1MEN1CASP1CASP7KMT2A
SCHEMBL29580973 0.77 CYP1A2 (0.46) ALDH1A1CYP1A2CYP3A4ACACB
SCHEMBL13046229 0.77 CYP1A2 (0.46) ALDH1A1CYP1A2CYP3A4ACACB
SCHEMBL28189564 0.76 NPC1 (0.58) ALDH1A1CASP1CYP1A2CYP2C19HTT
SCHEMBL2224500 0.76 CYP1A2 (0.50) CYP1A2
SCHEMBL1914269 0.76 CYP1A1 (0.38) CYP1A2GRM5
SCHEMBL6854251 0.75 ALDH1A1 (0.46) ALDH1A1MEN1CASP1CASP7KMT2A
SCHEMBL6878742 0.75 ALDH1A1 (0.53) ALDH1A1MEN1CASP1CASP7KMT2A
SCHEMBL740305 0.75 ALDH1A1 (0.53) ALDH1A1MEN1CASP1CASP7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739338-A SKIN DISORDERS, ANTIINFLAMMATORY AGENTS, ANTITUMOR AGENTS, VISION DEFECTS, VIRICIDES, IMMUNOSUPPRESSANTS ALLERGAN (US) 1998-04-14 US disclosed