SCHEMBL8615872

SCHEMBL8615872

CCCCC(C)c1cccc2c(NC(=N)NC=O)cc(-c3ccccc3)nc12

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 3/20 0.38
CACNA2D1 P54289 1/20 0.38
ACP1 P24666 1/20 0.37
ADORA1 P30542 4/20 0.36
MOK Q9UQ07 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 1/20 0.34
DHODH Q02127 1/20 0.34
ABCB1 P08183 1/20 0.34
ABCC1 P33527 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617418 0.94 ADORA1 (0.39) TACR3CACNA2D1ACP1ADORA1MOK
SCHEMBL8613769 0.91 ACP1 (0.39) TACR3CACNA2D1ACP1ADORA1MOK
SCHEMBL8614839 0.83 TACR3 (0.45) TACR3CACNA2D1ACP1MOKDHODH
SCHEMBL8615672 0.81 MOK (0.38) TACR3ACP1ADORA1MOKADORA3
SCHEMBL8620687 0.80 PDE10A (0.45) ACP1ADORA1ADORA2A
SCHEMBL8620939 0.80 ADORA1 (0.47) ADORA1ADORA3ADORA2A
SCHEMBL8613487 0.79 KDM4E (0.44) ACP1ABCB1ABCC1ABCG2
SCHEMBL8615997 0.78 CCR6 (0.45) ACP1ADORA3ABCB1ABCC1ABCG2
SCHEMBL8620923 0.78 ALOX5AP (0.38)
SCHEMBL8615114 0.78 ACP1 (0.36) CACNA2D1ACP1ADORA1MOKADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed