SCHEMBL8616655

SCHEMBL8616655

CCCCCCc1ccccc1-c1cc(NC(=N)NC=O)c2ccccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
GAA P10253 4/20 0.40
HPGD P15428 4/20 0.40
HSD17B10 Q99714 3/20 0.40
GLA P06280 3/20 0.40
TSHR P16473 2/20 0.40
MAPK1 P28482 1/20 0.40
PDE10A Q9Y233 1/20 0.40
DHODH Q02127 1/20 0.39
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
ACP1 P24666 3/20 0.38
POLB P06746 1/20 0.37
APOBEC3A P31941 1/20 0.37
HTT P42858 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618647 0.99 KDM4E (0.41) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8614301 0.97 PDE10A (0.42) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8613259 0.92 PDE10A (0.42) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8616287 0.89 PDE10A (0.49) PDE10AACP1HTTMOK
SCHEMBL8619516 0.85 PDE10A (0.44) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8614159 0.84 PDE10A (0.45) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8614071 0.83 PDE10A (0.40) KDM4EALDH1A1GAAGLAPDE10A
SCHEMBL8616012 0.83 PDE10A (0.40) KDM4EALDH1A1PDE10ADHODHMAPT
SCHEMBL8613965 0.83 PDE10A (0.46) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL8615672 0.82 MOK (0.38) PDE10ADHODHACP1MOK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed