SCHEMBL8614301

SCHEMBL8614301

CCCCc1ccccc1-c1cc(NC(=N)NC=O)c2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.42
DHODH Q02127 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GLA P06280 1/20 0.40
MAPK1 P28482 1/20 0.40
ACP1 P24666 3/20 0.40
MOK Q9UQ07 3/20 0.38
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
TRPV1 Q8NER1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618647 0.98 KDM4E (0.41) PDE10ADHODHKDM4EALDH1A1GAA
SCHEMBL8616655 0.97 KDM4E (0.40) PDE10ADHODHKDM4EALDH1A1GAA
SCHEMBL8613259 0.95 PDE10A (0.42) PDE10ADHODHKDM4EALDH1A1GAA
SCHEMBL8616287 0.92 PDE10A (0.49) PDE10AACP1MOKTRPV1
SCHEMBL8614071 0.86 PDE10A (0.40) PDE10AKDM4EALDH1A1GAAGLA
SCHEMBL8616012 0.86 PDE10A (0.40) PDE10ADHODHKDM4EALDH1A1ACP1
SCHEMBL8613965 0.85 PDE10A (0.46) PDE10ADHODHKDM4EALDH1A1GAA
SCHEMBL8614159 0.84 PDE10A (0.45) PDE10AKDM4EALDH1A1GAAHPGD
SCHEMBL8619516 0.84 PDE10A (0.44) PDE10ADHODHKDM4EALDH1A1GAA
SCHEMBL8620892 0.83 HTT (0.47) KDM4EALDH1A1HPGDACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed