SCHEMBL8617537

SCHEMBL8617537

N=C(NC=O)Nc1cc(-c2cccc(C(F)(F)F)c2)nc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 4/20 0.54
CA12 O43570 3/20 0.48
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
CA9 Q16790 3/20 0.48
ABCG2 Q9UNQ0 3/20 0.44
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44
KMO O15229 1/20 0.40
DHODH Q02127 1/20 0.40
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618214 0.89 ACP1 (0.53) ACP1ABCG2ABCB1ABCC1TRPV1
SCHEMBL8617753 0.87 ACP1 (0.51) ACP1ABCG2ABCB1ABCC1PDE10A
SCHEMBL8619429 0.86 ABCG2 (0.44) ACP1CA12CA1CA2CA9
SCHEMBL8615255 0.86 ABCG2 (0.53) ACP1ABCG2ABCB1ABCC1
SCHEMBL8617796 0.85 ACP1 (0.51) ACP1ABCG2ABCB1ABCC1MAPT
SCHEMBL8614861 0.85 AKR1C3 (0.53) ACP1ABCG2ABCB1ABCC1
SCHEMBL8615219 0.84 ABCG2 (0.42) ACP1ABCG2ABCB1ABCC1
SCHEMBL8614345 0.84 ABCG2 (0.44) ACP1ABCG2ABCB1ABCC1MAPT
SCHEMBL8614079 0.84 ACP1 (0.52) ACP1CA12CA1CA2CA9
SCHEMBL8618948 0.84 MEN1 (0.50) ACP1ABCG2ABCB1ABCC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed