SCHEMBL8614079

SCHEMBL8614079

N=C(NC=O)Nc1cc(-c2cccc(Cl)c2)nc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 11/20 0.52
ALDH1A1 P00352 1/20 0.49
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
GFER P55789 1/20 0.48
KMT2A Q03164 1/20 0.48
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
TACR3 P29371 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617753 0.90 ACP1 (0.51) ACP1MEN1GFERKMT2ASMN1; SMN2
SCHEMBL8619389 0.88 TACR3 (0.41) ACP1ALDH1A1CA12CA1CA2
SCHEMBL8614861 0.88 AKR1C3 (0.53) ACP1MEN1GFERKMT2AABCB1
SCHEMBL8615255 0.87 ABCG2 (0.53) ACP1ABCB1ABCC1ABCG2
SCHEMBL8614345 0.87 ABCG2 (0.44) ACP1ALDH1A1MEN1NPC1RAB9A
SCHEMBL8618948 0.87 MEN1 (0.50) ACP1ALDH1A1MEN1NPC1RAB9A
SCHEMBL8617812 0.86 MAPK1 (0.46) ACP1ALDH1A1MEN1KMT2ACA12
SCHEMBL8617537 0.84 ACP1 (0.54) ACP1CA12CA1CA2CA9
SCHEMBL8614857 0.84 ABCB1 (0.55) ACP1ALDH1A1MEN1NPC1RAB9A
SCHEMBL8619401 0.84 ABCB1 (0.44) ACP1ABCB1ABCC1ABCG2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed