SCHEMBL8617641

SCHEMBL8617641

O=C(NCCCCSc1ccccn1)c1ccccn1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.63
NPC1 O15118 3/20 0.60
RAB9A P51151 3/20 0.60
NFKB1 P19838 1/20 0.60
NFKB2 Q00653 1/20 0.60
RELA Q04206 1/20 0.60
HDAC3 O15379 1/20 0.59
HDAC4 P56524 1/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC7 Q8WUI4 1/20 0.59
HDAC2 Q92769 1/20 0.59
HDAC10 Q969S8 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HDAC9 Q9UKV0 1/20 0.59
HDAC5 Q9UQL6 1/20 0.59
ALDH1A1 P00352 2/20 0.56
KMT2A Q03164 6/20 0.56
MEN1 O00255 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618595 0.86 NPC1 (0.67) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8614872 0.85 KMT2A (0.57) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8966355 0.84 SMN1; SMN2 (0.60) SMN1; SMN2HDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8620230 0.84 KMT2A (0.56) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8620519 0.83 NPC1 (0.55) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8516755 0.82 SMN1; SMN2 (0.90) SMN1; SMN2HDAC3HDAC4HDAC1HDAC7
SCHEMBL8617471 0.82 NPC1 (0.68) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8619134 0.82 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
SCHEMBL8615169 0.81 KDM4E (0.58) SMN1; SMN2NPC1RAB9ANFKB1NFKB2
Hydrochloric Acid SCHEMBL8618623 0.81 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ANFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767121-A ANTIINFLAMMATORY AND -ARTHRITIC AGENTS; ANTIPYRETICS; ANALGESICS; ADHESION PROTEIN EXPRESSION AND CYCLOXYGENASE AND 5-LIPOXYGENASE INHIBITORS; IMMUNOSUPPRESSANTS AND -MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-16 US disclosed