SCHEMBL8618210

SCHEMBL8618210

N=C(N)NC(=O)c1cc(-c2ccc(C(F)(F)F)cc2)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RUVBL1 Q9Y265 1/20 0.56
TRPV1 Q8NER1 6/20 0.56
TACR3 P29371 5/20 0.53
CYP3A4 P08684 2/20 0.52
KDM4E B2RXH2 2/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
KMT2A Q03164 1/20 0.52
KCNH2 Q12809 1/20 0.52
CYP2C9 P11712 1/20 0.51
CA12 O43570 2/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA9 Q16790 2/20 0.51
NPC1 O15118 1/20 0.51
MAPT P10636 1/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617534 0.89 CA12 (0.64) RUVBL1TRPV1TACR3CYP3A4KDM4E
SCHEMBL8615804 0.89 KDM4E (0.64) RUVBL1TRPV1TACR3CYP3A4KDM4E
SCHEMBL8617743 0.88 CYP3A4 (0.65) TACR3CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8614006 0.87 KDM4E (0.60) TACR3CYP3A4KDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8620745 0.87 CYP3A4 (0.64) TACR3CYP3A4KDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8620121 0.86 KDM4E (0.59) TACR3CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8620931 0.86 POLB (0.66) TACR3CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8615244 0.86 CYP3A4 (0.56) TACR3CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8616671 0.86 TRPV1 (0.55) RUVBL1TRPV1TACR3CYP3A4KDM4E
SCHEMBL8617544 0.85 MEN1 (0.60) TACR3CYP3A4KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed