SCHEMBL8616671

SCHEMBL8616671

N=C(N)NC(=O)c1cc(-c2ccc(OC(F)(F)F)cc2)nc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.55
RUVBL1 Q9Y265 1/20 0.53
ACP1 P24666 1/20 0.53
DHODH Q02127 1/20 0.53
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
TACR3 P29371 4/20 0.51
CYP3A4 P08684 2/20 0.50
KLK7 P49862 1/20 0.50
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
KCNH2 Q12809 1/20 0.49
MAPT P10636 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
GLA P06280 1/20 0.48
GAA P10253 1/20 0.48
ATM Q13315 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617790 0.90 KDM4E (0.54) TRPV1DHODHMEN1KMT2ATACR3
SCHEMBL8620708 0.86 MEN1 (0.68) RUVBL1MEN1KMT2ARAB9ANPC1
SCHEMBL8618210 0.86 RUVBL1 (0.56) TRPV1RUVBL1DHODHMEN1KMT2A
SCHEMBL8617743 0.85 CYP3A4 (0.65) DHODHMEN1KMT2ATACR3CYP3A4
SCHEMBL8614006 0.85 KDM4E (0.60) DHODHMEN1KMT2ARAB9ANPC1
Hydrochloric Acid SCHEMBL8620745 0.84 CYP3A4 (0.64) DHODHMEN1KMT2ATACR3CYP3A4
Hydrochloric Acid SCHEMBL8620121 0.84 KDM4E (0.59) DHODHMEN1KMT2ARAB9ANPC1
SCHEMBL8620931 0.83 POLB (0.66) DHODHMEN1KMT2ATACR3CYP3A4
SCHEMBL8615244 0.83 CYP3A4 (0.56) DHODHMEN1KMT2ATACR3CYP3A4
SCHEMBL8613377 0.83 TACR3 (0.48) MEN1KMT2ATACR3CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed