SCHEMBL8618936

SCHEMBL8618936

Cc1cc(C)cc(-c2cc(C(=O)NC(=N)N)c3ccccc3n2)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.56
MEN1 O00255 9/20 0.53
KMT2A Q03164 9/20 0.53
ALDH1A1 P00352 5/20 0.53
CYP1A2 P05177 2/20 0.53
ALOX12 P18054 2/20 0.53
CYP2C19 P33261 2/20 0.53
KCNH2 Q12809 2/20 0.53
PTGER4 P35408 2/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 2/20 0.52
KDM4E B2RXH2 2/20 0.52
MAPT P10636 3/20 0.52
LMNA P02545 3/20 0.52
HTT P42858 1/20 0.52
TACR3 P29371 4/20 0.51
CNR1 P21554 1/20 0.51
GPR55 Q9Y2T6 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618943 0.91 MEN1 (0.65) CYP3A4MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8615354 0.91 CYP3A4 (0.65) CYP3A4MEN1KMT2AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8613665 0.90 MEN1 (0.64) CYP3A4MEN1KMT2AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8618111 0.89 CYP3A4 (0.64) CYP3A4MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8617743 0.89 CYP3A4 (0.65) CYP3A4MEN1KMT2AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8620745 0.88 CYP3A4 (0.64) CYP3A4MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8618197 0.87 ALDH1A1 (0.49) CYP3A4MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8615244 0.87 CYP3A4 (0.56) CYP3A4MEN1KMT2AALDH1A1KCNH2
SCHEMBL8618148 0.86 TP53 (0.65) CYP3A4MEN1KMT2AALDH1A1CYP1A2
SCHEMBL8615674 0.85 CYP3A4 (0.58) CYP3A4MEN1KMT2AALDH1A1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed