SCHEMBL8620388

SCHEMBL8620388

CCOc1cnc(-c2ccc(CCC(C)OC(C)=O)cc2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 13/20 0.44
MMP12 P39900 1/20 0.41
ADORA3 P0DMS8 1/20 0.39
MAPT P10636 2/20 0.39
THRB P10828 1/20 0.39
ACACA Q13085 5/20 0.38
FFAR1 O14842 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
RARB P10826 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864496 0.89 RARB (0.46) ACACBMAPTRARBKDM4EMEN1
SCHEMBL9096988 0.83 RARB (0.47) ACACBMAPTRARBKDM4EMEN1
SCHEMBL8620927 0.83 MAPT (0.40) ACACBMAPTTHRBFFAR1FFAR4
SCHEMBL9096672 0.82 RARB (0.49) ACACBMAPTRARBKDM4EMEN1
SCHEMBL9095535 0.82 RARB (0.49) ACACBMAPTRARBKDM4EMEN1
SCHEMBL8593405 0.80 CNR1 (0.38) ACACBMMP12MAPTTHRBRARB
SCHEMBL8593408 0.80 CNR1 (0.38) ACACBMMP12MAPTTHRBRARB
SCHEMBL8591411 0.80 RARB (0.40) MAPTTHRBPPARARARBKDM4E
SCHEMBL8594480 0.80 RARB (0.40) MAPTTHRBPPARARARBKDM4E
SCHEMBL8593933 0.80 RARB (0.40) MAPTTHRBPPARARARBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537620-B1 Nitrogen-containing heterorings ROLIC AG (CH) 1998-01-07 EP disclosed
US-5326497-A Nitrogen heterocycles and liquid crystalline mixtures containing them HOFFMANN-LA ROCHE INC. (US) 1994-07-05 US disclosed
EP-0537620-A1 Nitrogen-containing heterorings F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed